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ַ > Ϲݰַ 21
Խù 66,690, ֱ 254
ǰ塼rd17.cia158.comƱ ĬŸ
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Ʊ ߱ ظü Ͽ cGMP ؽŰ 5 ̿(phosphodiesterase) ȿҸ μ ظü Ǵ ȭ (NO) ۿ ȭϿ Ƶ Ȯ ӽŴμ ߱ ġȿ δ.
Ʊ Ȯ Ű ȯ ġϴ ̾. 嵥 ƿ ġ ⺸ٴ ƿ ġ Ǵ . ̰ ü Ʋ ư پִ ̱ ε, 忡 ܼ ȮDZ⸸ ̾, ư پִٺ, ȮǸ ݴη ٽ ư , ̰ ߱⸦ ִ ̴.
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<߱ ġ> 汸 ߱ġ Ʊ ּ ǵ̸, cGMP-Ư Ͷ 5 (PDE 5) Դϴ. ǵ ȭи 1-[[3-(6,7-dihydro-1-methyl-7-oxo-3-propyl-1H-pyrazolo[4,3- d]pyrimidin-5-yl)-4-ethoxyphenyl]sulfonyl]-4-methylpiperazine citrate ̸ ϴ. ǵ и̸ 3.5 mg/ml 뼺 ڷ 666.7 Դϴ. Ʊ( ǵ) ణ ձ ̾Ƹ Ǫ ʸ, ǵ 25mg, 50mg, 100mg شϴ ǵ () 35.11 mg, 70.23 mg, 140.45mg 3 뷮 汸 㰡Ǿ ֽϴ.
߱ ġ ó ȿ ̾ 찡 ִ. ̷ 뷮 øų ٸ ٲ Ѵٰ , Ծ Ȯغ ʿ䰡 ִ. ߱ ġ ð Ծ, Ǵ Ļ Ŀ ߴ, ų ⸧ ⸦ Ծ ü ȿ ִ. Ʊ, ȡ ǵ ӿ Ծ Ѵ. Ʊ ӿ ϸ 30 ߱ ȿ Ÿ , 30~120 ̿ ִ ߱ Ÿ. ౹ 30~60 ϶ ϰ ִ. ݴ Ŀ Ʊ 90 ̻ ִ ߱ ȿ Ÿ. 谡 ߱ 1ð 踦 õ ߱Ⱑ ʾƼ , ȿ ١ ִ. 90~120 ȿ Ÿٰ ϴ, ӿ ϸ ߱ 30% ɼ ũ. ̷ Ļ ⸧ ε巯. Ư Ļ Ŀ ߱ ϸ ȿ ʰ ǰų ִ. , ȿ ʹٸ ȿ 빰 ӿ ؾ Ѵٴ ˾Ƶ ʿ䰡 ִ. Ŀ ߱ ġδ ٵ е ִ. ǰ ϶. ϶ ϸ ִ ȿ 60 ߰ ǰ, ִ ȿ 18% Ѵ. Ÿٶ þ˸ ⺻ Ư 2ð ؾ ȿ ִ ̴. İ Բ ص ȿ ̰ , 1ð ̳ ȿ ϴ. 2ð ־ ȿ ִ. ٸ ӿ ߱ ġ ؾ ִ. ӿ ϸ ȿŭ ۿ뵵 ϰ Ÿ. Ʊ, , ϶ ǵŸ, ٵ ġ , Ϸ , ȭҷ, þ 帲 Ÿ 忡 δ ִ. ߱ ġ Ȯ ִ ε, ƴ϶ Ȯ Ͻ Ѵ. ¸ ȮǸ Ͻ ų ȭ ǰ, Ȯ ؾ ϴ 忡 δ ִ. ϴ ȣ ΰϰ ν þ ̻ ۿ Ÿ Ѵ. ߱ ġ ۿ ӿ ۿ뵵 ϰ Ÿ ݸ, ۿ ʰ ߵ 쿡 ӿ ص ũ ʴ´. Ÿٶ þ˸ Ļ ο ۿ ϰ Ÿ. Ÿٶ ۿ , ̴. 3 ӵ ִ. ̿ܿ ۿ ϰ Ÿ ̴. Ÿٶ ȿ Ⱑ 36ð ȿ Ǵ ̶ ۿ뵵 Ÿ. ó ʿ Ʊ Ʊ Ʊ ı Ʊ Ʈ Ʊ ȵǴ Ʊ Ʊ Ʊ ó¹
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